SCHEMBL7826319

SCHEMBL7826319

COc1cccc2c(N3CCc4cccc(C)c4C3C)nc(Cl)nc12

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 3/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
RAD52 P43351 1/20 0.39
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.35
HTR1A P08908 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811938 0.86 ADORA2A (0.42) KDM4EGLAGAAHTTALDH1A1
SCHEMBL7821140 0.86 ADORA2A (0.42) KDM4EGLAGAAHTTALDH1A1
SCHEMBL7811946 0.86 ADORA2A (0.42) KDM4EGLAGAAHTTALDH1A1
SCHEMBL7822272 0.84 KDM4E (0.38) KDM4EGLAGAAHTTALDH1A1
SCHEMBL7818228 0.84 KDM4E (0.39) KDM4EGLAGAAHTTALDH1A1
SCHEMBL7810634 0.81 TP53 (0.40) KDM4ELMNARAD52HPGD
Hydrochloric Acid SCHEMBL7826307 0.80 RAD52 (0.41) KDM4EHTTLMNARAD52HPGD
SCHEMBL7819071 0.79 MAP4K1 (0.38)
Hydrochloric Acid SCHEMBL7825400 0.78 MAP4K1 (0.37)
SCHEMBL7820129 0.78 ADORA2A (0.40) KDM4EGLAGAAHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677049-B1 QUINAZOLINE DERIVATIVES YUHAN CORP LTD (KR) 2001-07-25 EP disclosed
US-5686458-A Quinazoline deriviates for treating peptic ulcer YUHAN CORPORATION (KR) 1997-11-11 US disclosed
EP-0677049-A1 QUINAZOLINE DERIVATIVES YUHAN CORPORATION, LTD. (KR) 1995-10-18 EP disclosed
WO-1994014795-A1 QUINAZOLINE DERIVATIVES YUHAN CORPORATION (KR) 1994-07-07 WO disclosed