SCHEMBL7821140

SCHEMBL7821140

COc1cccc2c(N3CCc4ccccc4[C@@H]3C)nc(Cl)nc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.42
KDM4E B2RXH2 4/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 4/20 0.38
DRD1 P21728 3/20 0.37
LMNA P02545 2/20 0.37
NPC1 O15118 1/20 0.37
RAD52 P43351 1/20 0.37
DRD2 P14416 1/20 0.37
DRD5 P21918 1/20 0.37
DRD3 P35462 1/20 0.37
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811946 1.00 ADORA2A (0.42) ADORA2AKDM4EGLAGAAHTT
SCHEMBL7811938 1.00 ADORA2A (0.42) ADORA2AKDM4EGLAGAAHTT
SCHEMBL7818228 0.89 KDM4E (0.39) KDM4EGLAGAAHTTALDH1A1
SCHEMBL7820129 0.87 ADORA2A (0.40) ADORA2AKDM4EGLAGAAHTT
SCHEMBL7820068 0.87 KDM4E (0.39) ADORA2AKDM4EGLAGAAHTT
SCHEMBL7810515 0.87 KDM4E (0.39) ADORA2AKDM4EGLAGAAHTT
SCHEMBL7826319 0.86 KDM4E (0.40) KDM4EGLAGAAHTTALDH1A1
SCHEMBL7818704 0.86 KDM4E (0.38) ADORA2AKDM4EGLAGAAHTT
SCHEMBL7820223 0.84 KDM4E (0.38) ADORA2AKDM4EGLAGAAHTT
SCHEMBL7818490 0.83 EHMT2 (0.40) ADORA2AKDM4EGLAGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677049-B1 QUINAZOLINE DERIVATIVES YUHAN CORP LTD (KR) 2001-07-25 EP disclosed
US-5686458-A Quinazoline deriviates for treating peptic ulcer YUHAN CORPORATION (KR) 1997-11-11 US disclosed
EP-0677049-A1 QUINAZOLINE DERIVATIVES YUHAN CORPORATION, LTD. (KR) 1995-10-18 EP disclosed
WO-1994014795-A1 QUINAZOLINE DERIVATIVES YUHAN CORPORATION (KR) 1994-07-07 WO disclosed