SCHEMBL7826641

SCHEMBL7826641

Fc1cccc(Cc2cc(Br)cs2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
TAAR1 Q96RJ0 3/20 0.42
IDO1 P14902 2/20 0.41
AGXT P21549 2/20 0.41
DAO P14920 1/20 0.40
PRNP P04156 2/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
MIF P14174 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28571991 0.79 MAPK1 (0.56) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL12651459 0.77 KDM4E (0.51) KDM4ETAAR1
SCHEMBL7825397 0.76 TAAR1 (0.42) MAOBMEN1KMT2AKDM4EALDH1A1
SCHEMBL3300303 0.74 TAAR1 (0.60) MAOBALDH1A1TAAR1IDO1AGXT
SCHEMBL23011377 0.73 MAOB (0.47) MAOBALDH1A1TAAR1IDO1AGXT
SCHEMBL28567520 0.70 SLC6A4 (0.40) HPGDTAAR1IDO1DAOMGAM
SCHEMBL156072 0.70 TAAR1 (0.44) MAOBTAAR1IDO1AGXT
SCHEMBL153073 0.69 MAPT (0.36) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL21205126 0.69 MEN1 (0.47) MAOBMEN1KMT2AKDM4EALDH1A1
SCHEMBL919866 0.69 P2RX7 (0.43) MEN1KMT2AKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086091-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2001-10-10 EP disclosed
US-6262055-B1 SULFUR-CONTAINING HETEROARYL DIOXO-BUTYRIC ACID DERIVATIVES MERCK & CO., INC. 2001-07-17 US disclosed
EP-1086091-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2001-03-28 EP disclosed
WO-1999062897-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed