SCHEMBL7828301

SCHEMBL7828301

CC(=O)c1cccc([N+](=O)[O-])c1.CN(C)S(=O)(=O)n1cnc(C(C)(O)c2cccc([N+](=O)[O-])c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
MAOB P27338 1/20 0.38
PTPRC P08575 1/20 0.38
RAB9A P51151 3/20 0.37
MAPT P10636 3/20 0.37
HTT P42858 2/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
NPC1 O15118 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
RECQL P46063 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
SLC6A9 P48067 1/20 0.36
SLC6A5 Q9Y345 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7101212 0.92 PTPRC (0.44) ALDH1A1PTPRCMAPTHTTKMT2A
SCHEMBL7100834 0.76 ALDH1A1 (0.45) ALDH1A1RAB9AMAPTHTTKMT2A
SCHEMBL7100881 0.74 ALDH1A1 (0.41) ALDH1A1RAB9AMAPTHTTKMT2A
SCHEMBL7100864 0.70 MAPT (0.39) ALDH1A1RAB9AMAPTHTTKMT2A
SCHEMBL7100873 0.70 MAPT (0.39) ALDH1A1RAB9AMAPTHTTKMT2A
SCHEMBL54610 0.69 ALDH1A1 (1.00) ALDH1A1MAOBRAB9AMAPTHTT
SCHEMBL30780024 0.69 ALDH1A1 (1.00) ALDH1A1MAOBRAB9AMAPTHTT
SCHEMBL7100452 0.68 KMT2A (0.44) ALDH1A1RAB9AMAPTHTTKMT2A
SCHEMBL28042240 0.68 ALDH1A1 (0.96) ALDH1A1MAOBRAB9AMAPTHTT
Hydrochloric Acid SCHEMBL27577695 0.68 ALDH1A1 (0.96) ALDH1A1MAOBRAB9AMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102754-A1 IMIDAZOLES AND RELATED COMPOUNDS AS ALPHA-1A AGONISTS ABBOTT LABORATORIES (US) 2001-05-30 EP disclosed
WO-2000007997-A1 IMIDAZOLES AND RELATED COMPOUNDS AS α1A AGONISTS ABBOTT LABORATORIES (US) 2000-02-17 WO disclosed