SCHEMBL7828429

SCHEMBL7828429

C=CCN(CC=C)c1ccc(C(=O)CC(=O)C(=O)O)s1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 13/20 0.48
ERCC5 P28715 12/20 0.48
RNASEH1 O60930 1/20 0.44
PTPN1 P18031 4/20 0.37
TYMS P04818 1/20 0.34
HAO1 Q9UJM8 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7818173 0.78 FEN1 (0.52) FEN1ERCC5RNASEH1PTPN1TYMS
SCHEMBL7828343 0.77 GSK3B (0.42) TYMS
SCHEMBL7818129 0.77 ERCC5 (0.55) FEN1ERCC5RNASEH1PTPN1HAO1
SCHEMBL7828436 0.74 ERCC5 (0.48) FEN1ERCC5RNASEH1PTPN1
SCHEMBL7818280 0.69 ERCC5 (0.52) FEN1ERCC5RNASEH1PTPN1HAO1
SCHEMBL11211936 0.69 DAO (0.36) TYMS
SCHEMBL7829542 0.65 ERCC5 (0.47) FEN1ERCC5RNASEH1
SCHEMBL5772644 0.63 ERCC5 (0.44) FEN1ERCC5RNASEH1
SCHEMBL7830529 0.63 ERCC5 (0.59) FEN1ERCC5RNASEH1PTPN1HAO1
SCHEMBL7828353 0.62 ERCC5 (0.57) FEN1ERCC5RNASEH1PTPN1HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086091-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2001-10-10 EP claimed
US-6262055-B1 SULFUR-CONTAINING HETEROARYL DIOXO-BUTYRIC ACID DERIVATIVES MERCK & CO., INC. 2001-07-17 US claimed
EP-1086091-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2001-03-28 EP claimed
WO-1999062897-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1086091-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2001-10-10 EP disclosed
US-6262055-B1 SULFUR-CONTAINING HETEROARYL DIOXO-BUTYRIC ACID DERIVATIVES MERCK & CO., INC. 2001-07-17 US disclosed
EP-1086091-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2001-03-28 EP disclosed
WO-1999062897-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed