SCHEMBL7828530

SCHEMBL7828530

O=C(O)CCc1nc(-c2cccc3ccccc23)no1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.64
HPGD P15428 4/20 0.64
CYP3A4 P08684 1/20 0.64
MCL1 Q07820 1/20 0.55
TSHR P16473 4/20 0.54
ATM Q13315 3/20 0.51
LMNA P02545 3/20 0.51
FFAR1 O14842 2/20 0.50
TP53 P04637 3/20 0.49
MITF O75030 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49
S1PR1 P21453 1/20 0.47
MAPT P10636 2/20 0.47
MAPK1 P28482 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
KDM4E B2RXH2 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6325690 0.83 ALDH1A1 (0.67) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL6326180 0.82 HPGD (0.65) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL6332414 0.82 ALDH1A1 (0.65) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL6328228 0.82 ALDH1A1 (0.65) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL6326021 0.82 ATM (0.72) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL6326409 0.81 ALDH1A1 (0.60) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL6332427 0.80 TSHR (0.60) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL5330405 0.80 ALDH1A1 (0.83) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL7837661 0.79 ALDH1A1 (0.55) ALDH1A1HPGDCYP3A4MCL1TSHR
SCHEMBL6327192 0.79 ALDH1A1 (0.61) ALDH1A1HPGDCYP3A4MCL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329389-B1 HETEROCYCLIC AMINES AND DERIVATIVES, SOMATOSTATIN AND ANTIDIABETIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-12-11 US disclosed
EP-1070054-A1 AMINE COMPOUNDS, THEIR PRODUCTION AND THEIR USE AS SOMATOSTATIN RECEPTOR ANTAGONISTS OR AGONISTS Takeda Chemical Industries, Ltd. (JP) 2001-01-24 EP disclosed
WO-1999052875-A1 AMINE COMPOUNDS, THEIR PRODUCTION AND THEIR USE AS SOMATOSTATIN RECEPTOR ANTAGONISTS OR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-21 WO disclosed