SCHEMBL7829615

SCHEMBL7829615

Cc1cc(=O)oc2c(C)c3c(cc12)CC(CN1CCOCC1)O3

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
ATM Q13315 1/20 0.47
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TP53 P04637 1/20 0.43
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
HTR1A P08908 2/20 0.40
HTR2A P28223 1/20 0.40
KDM4E B2RXH2 3/20 0.40
POLB P06746 1/20 0.40
PRKDC P78527 1/20 0.40
KCNA3 P22001 1/20 0.39
PTPN1 P18031 1/20 0.39
P2RY12 Q9H244 1/20 0.38
ALDH1A1 P00352 2/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7814575 0.84 KMT2A (0.38) KMT2AATMTP53PDE3BPDE3A
SCHEMBL7946011 0.83 KDM4E (0.49) KMT2AHSD17B10KDM4EPOLBALDH1A1
SCHEMBL7822499 0.82 MAOA (0.43) KMT2AATMCASP1CASP7HSD17B10
SCHEMBL7483011 0.80 MAOA (0.43) KMT2AATMCASP1CASP7HSD17B10
SCHEMBL7822484 0.78 MCL1 (0.41) KMT2ACASP1CASP7HSD17B10KDM4E
SCHEMBL7825702 0.77 MAOA (0.40) KMT2AATMCASP1CASP7HSD17B10
SCHEMBL7822726 0.77 MAOA (0.40) KMT2ACASP1CASP7HSD17B10KDM4E
Iodide SCHEMBL7487937 0.77 MCL1 (0.41) KMT2ACASP1CASP7HSD17B10KDM4E
SCHEMBL9134783 0.76 MAOA (0.46) KMT2ACASP1CASP7HSD17B10TP53
SCHEMBL11320599 0.74 MAOB (0.46) KMT2ACASP1CASP7HSD17B10TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133498-A2 AMINO-AND MERCURIO-SUBSTITUTED 4', 5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2001-09-19 EP disclosed
US-6255324-B1 MICROBIOCIDES; SKIN DISORDERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2001-07-03 US disclosed
WO-2000031081-A2 AMINO- AND MERCURIO-SUBSTITUTED 4',5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2000-06-02 WO disclosed