SCHEMBL7832085

SCHEMBL7832085

Nc1cc(-c2ccoc2)ccc1Nc1cccc(-n2ccnc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 0.42
CYP3A4 P08684 9/20 0.42
CYP2D6 P10635 9/20 0.42
CYP2C19 P33261 8/20 0.42
LMNA P02545 5/20 0.42
ALDH1A1 P00352 4/20 0.42
CLK4 Q9HAZ1 4/20 0.42
TP53 P04637 2/20 0.42
HSD17B10 Q99714 5/20 0.38
TDP1 Q9NUW8 5/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
HDAC1 Q13547 2/20 0.37
MAPK1 P28482 5/20 0.35
ALOX15 P16050 3/20 0.35
USP2 O75604 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834399 0.83 CYP1A2 (0.49) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL7830304 0.83 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL7829252 0.80 ABL1 (0.46) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL2643607 0.70 HDAC2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL7831832 0.67 CYP1A2 (0.45) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL2643659 0.66 HDAC2 (0.43) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL9071943 0.66 HDAC2 (0.41) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL2643656 0.66 HDAC2 (0.41) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL2643742 0.65 MAP4K4 (0.42) CYP1A2CYP3A4CYP2D6CYP2C19LMNA
SCHEMBL2643125 0.65 SYK (0.37) CYP1A2CYP3A4CYP2D6CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1164134-A1 Benzimidazole compounds and their use as modulators of the GABA A receptor complex NEUROSEARCH A/S (DK) 2001-12-19 EP disclosed
EP-0821684-B1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABA A? RECEPTOR COMPLEX NEUROSEARCH AS (DK) 2001-12-05 EP disclosed
US-5922724-A Benzimidazole compounds and their use as modulators of the GABA a receptor complex NEUROSEARCH A/S (DK) 1999-07-13 US disclosed