SCHEMBL7832807

SCHEMBL7832807

CCOc1cccc(OCC)c1N(C)Cc1nc2cc(-n3ccnc3)ccc2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.38
F9 P00740 1/20 0.38
MAOA P21397 3/20 0.38
MAOB P27338 3/20 0.38
DRD4 P21917 1/20 0.37
CYP1A2 P05177 4/20 0.36
CYP2D6 P10635 4/20 0.36
CYP2C9 P11712 4/20 0.36
CYP2C19 P33261 4/20 0.36
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
CYP19A1 P11511 2/20 0.36
CYP3A4 P08684 3/20 0.36
FGFR1 P11362 1/20 0.35
FLT1 P17948 1/20 0.35
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7832812 0.92 CBFB (0.48) CBFBNCOA3F9MAOAMAOB
SCHEMBL7822322 0.90 MAOA (0.45) CBFBNCOA3F9MAOAMAOB
SCHEMBL7830531 0.85 MAOA (0.43) CBFBNCOA3F9MAOAMAOB
SCHEMBL7832658 0.84 NPC1 (0.40) CBFBNCOA3F9MAOAMAOB
SCHEMBL7832837 0.84 MAOA (0.42) CBFBNCOA3F9MAOAMAOB
SCHEMBL7833055 0.84 F9 (0.42) CBFBNCOA3F9MAOAMAOB
SCHEMBL7833472 0.83 CBFB (0.39) CBFBNCOA3F9MAOAMAOB
SCHEMBL7831669 0.83 F9 (0.40) CBFBNCOA3F9MAOAMAOB
SCHEMBL7822325 0.82 MAOA (0.48) CBFBNCOA3F9MAOAMAOB
SCHEMBL7833749 0.81 MEN1 (0.46) CBFBNCOA3F9MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
US-6040327-A INHIBITORS OF INTERLEUKINS; TREATING RHEUMATOID ARTHRITIS OR ARTHROSIS ADIR ET COMPAGNIE (FR) 2000-03-21 US disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed