SCHEMBL7833229

SCHEMBL7833229

O=C1C(=O)N(CCCl)c2ccc(F)cc21

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARK7 Q99497 5/20 0.67
NSD2 O96028 1/20 0.60
CHRM5 P08912 2/20 0.58
ALDH1A1 P00352 5/20 0.52
ALDH3A1 P30838 5/20 0.52
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA9 Q16790 2/20 0.50
ALDH2 P05091 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11150483 0.91 PARK7 (0.63) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL28909405 0.90 PARK7 (0.75) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL28547209 0.87 PARK7 (0.71) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL28546572 0.85 PARK7 (0.69) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL28533459 0.85 PARK7 (0.69) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL28539851 0.85 PARK7 (0.69) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL28547202 0.85 PARK7 (0.69) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL28533382 0.83 PARK7 (0.65) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL11149802 0.80 PARK7 (0.62) PARK7NSD2CHRM5ALDH1A1ALDH3A1
SCHEMBL20254404 0.80 PARK7 (1.00) PARK7NSD2CHRM5ALDH1A1ALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780388-B1 5HT1Dalpha and 5HT2A ligands LILLY CO ELI (GB) 2001-08-16 EP disclosed
US-6166040-A Indole compounds ELI LILLY AND COMPANY LIMITED (GB) 2000-12-26 US disclosed
EP-0963983-A1 Indol-2-ones as serotonin modulators ELI LILLY AND COMPANY LIMITED (GB) 1999-12-15 EP disclosed
WO-1999058525-A1 INDOLE DERIVATIVES AS 5-HT2A LIGANDS AND AS SEROTONINE REUPTAKE INHIBITORS ELI LILLY AND COMPANY LIMITED (GB) 1999-11-18 WO disclosed
US-5773448-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY LIMITED (GB) 1998-06-30 US disclosed
EP-0780388-A1 5HT1Dalpha and 5HT2A ligands LILLY INDUSTRIES LIMITED (GB) 1997-06-25 EP disclosed