SCHEMBL7833485

SCHEMBL7833485

CC(Oc1ccc(CC2SC(=O)NC2=O)cc1)c1nc2cnccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARG P37231 14/20 0.46
FFAR1 O14842 4/20 0.45
PPARA Q07869 3/20 0.45
CYP3A4 P08684 2/20 0.43
RXRA P19793 1/20 0.43
MPC2 O95563 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2C9 P11712 1/20 0.43
MAPT P10636 2/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1130956 0.87 FFAR1 (0.54) PPARGFFAR1PPARAMEN1TP53
SCHEMBL6896704 0.85 PPARG (0.51) PPARGFFAR1PPARAMPC2CYP2C8
Hydrochloric Acid SCHEMBL4177074 0.84 PPARG (0.51) PPARGFFAR1PPARACYP3A4RXRA
SCHEMBL6544205 0.84 PPARG (0.42) PPARGFFAR1PPARAMPC2CYP2C8
Hydrochloric Acid SCHEMBL6544229 0.83 PPARG (0.42) PPARGFFAR1PPARACYP3A4RXRA
SCHEMBL1130792 0.83 PPARG (0.54) PPARGFFAR1PPARAMPC2CYP2C8
Hydrochloric Acid SCHEMBL4165069 0.82 PPARG (0.53) PPARGFFAR1PPARACYP3A4RXRA
Hydrochloric Acid SCHEMBL6064786 0.82 PPARG (0.53) PPARGFFAR1PPARACYP3A4RXRA
SCHEMBL7243299 0.82 FFAR1 (0.49) PPARGFFAR1PPARACYP3A4MAPT
Hydrochloric Acid SCHEMBL6701459 0.82 PPARG (0.47) PPARGFFAR1PPARACYP3A4RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676398-B1 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO CO (JP) 2001-10-24 EP disclosed
US-6117893-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 2000-09-12 US disclosed
EP-1022274-A1 Oxazolidinedione and Thiazolidinedione derivatves, their preparation and their use Sankyo Company Limited (JP) 2000-07-26 EP disclosed
US-5977365-A HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
US-5962470-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 1999-10-05 US disclosed
US-5834501-A TREATING DIABETES OR HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 1998-11-10 US disclosed
US-5739345-A HYPOGLYCEMIC AND ANTIDIABETIC AGENTS SANKYO COMPANY, LIMITED (JP) 1998-04-14 US disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed