Carbutamide

Carbutamide

SCHEMBL7833740

CCCCNC(=O)NS(=O)(=O)c1ccc(N)cc1.Cc1cc(S(=O)(=O)O)ccc1N

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.61
ALDH1A1 P00352 2/20 0.61
LMNA P02545 2/20 0.61
TSHR P16473 2/20 0.61
ALB P02768 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
FBP1 P09467 11/20 0.54
CYP3A4 P08684 1/20 0.47
THRB P10828 1/20 0.47
NFKB1 P19838 1/20 0.47
HTR2A P28223 1/20 0.47
CYP2C19 P33261 1/20 0.47
ADRA1A P35348 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TBXA2R P21731 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbutamide SCHEMBL4078762 0.86 ALDH1A1 (0.76) CYP2C9ALDH1A1LMNATSHRALB
Carbutamide SCHEMBL49231 0.86 ALDH1A1 (0.76) CYP2C9ALDH1A1LMNATSHRALB
Carbutamide SCHEMBL7615910 0.78 ALDH1A1 (0.78) CYP2C9ALDH1A1LMNATSHRALB
Tolbutamide SCHEMBL15918 0.77 ALDH1A1 (1.00) CYP2C9ALDH1A1LMNATSHRALB
Tolbutamide SCHEMBL1536920 0.77 ALDH1A1 (1.00) CYP2C9ALDH1A1LMNATSHRALB
SCHEMBL8672470 0.76 ALDH1A1 (0.91) CYP2C9ALDH1A1LMNATSHRALB
Tolbutamide SCHEMBL11356450 0.76 ALDH1A1 (0.97) CYP2C9ALDH1A1LMNATSHRALB
Tolbutamide SCHEMBL4367531 0.76 ALDH1A1 (0.97) CYP2C9ALDH1A1LMNATSHRALB
Tolbutamide SCHEMBL11357518 0.76 ALDH1A1 (0.97) CYP2C9ALDH1A1LMNATSHRALB
Tolbutamide SCHEMBL140363 0.76 ALDH1A1 (0.97) CYP2C9ALDH1A1LMNATSHRALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946556-A4 COMBINATORIAL PROCESS FOR PREPARING HYDROFUROQUINOLINE LIBRARIES LILLY CO ELI (US) 2001-07-04 EP disclosed
EP-0946556-A1 COMBINATORIAL PROCESS FOR PREPARING HYDROFUROQUINOLINE LIBRARIES ELI LILLY AND COMPANY (US) 1999-10-06 EP disclosed
WO-1998027093-A1 COMBINATORIAL PROCESS FOR PREPARING HYDROFUROQUINOLINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-06-25 WO disclosed