SCHEMBL7834007

SCHEMBL7834007

CN(C)C(=O)Nc1snc(OCc2cccc(F)c2)c1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.44
MAOB P27338 6/20 0.41
PPIF P30405 1/20 0.39
ACVR2A P27037 1/20 0.39
TGFBR2 P37173 1/20 0.39
ANO1 Q5XXA6 2/20 0.39
DHODH Q02127 1/20 0.39
GRM5 P41594 2/20 0.39
PPARA Q07869 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
MAOA P21397 1/20 0.39
PARP10 Q53GL7 1/20 0.38
ALKBH1 Q13686 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3086638 0.91 ACVR2A (0.48) NR4A2MAOBPPIFACVR2ATGFBR2
SCHEMBL7832129 0.88 PPARG (0.42) NR4A2ACVR2ATGFBR2ALKBH1
SCHEMBL7830755 0.81 TSHR (0.41) NR4A2MAOBACVR2ATGFBR2MRGPRX4
SCHEMBL7832071 0.80 POLB (0.44) ACVR2ATGFBR2ANO1PPARAALKBH1
SCHEMBL3084724 0.80 ACVR2A (0.44) MAOBACVR2ATGFBR2PARP10
SCHEMBL3078380 0.80 ACVR2A (0.50) ACVR2ATGFBR2PARP10
SCHEMBL3082256 0.80 ACVR2A (0.49) MAOBACVR2ATGFBR2
SCHEMBL3078483 0.79 ACVR2A (0.48) MAOBACVR2ATGFBR2MAOAPARP10
SCHEMBL3091467 0.79 ACVR2A (0.48) ACVR2ATGFBR2ANO1
SCHEMBL3081929 0.79 ACVR2A (0.48) MAOBACVR2ATGFBR2GRM5MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084114-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2001-03-21 EP disclosed
WO-1999062890-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-12-09 WO disclosed