SCHEMBL7834255

SCHEMBL7834255

COc1ccnc(-c2ccc(F)c(N=C(N)N)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 4/20 0.56
CCR1 P32246 1/20 0.47
CCR5 P51681 1/20 0.47
CCR8 P51685 1/20 0.47
ATP4A P20648 5/20 0.43
ATP4B P51164 5/20 0.43
MAPT P10636 4/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
HTR3E A5X5Y0 2/20 0.38
HTR3B O95264 2/20 0.38
HTR3A P46098 2/20 0.38
HTR3D Q70Z44 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7239803 0.99 PLAU (0.55) PLAUCCR1CCR5CCR8ATP4A
Hydrochloric Acid SCHEMBL7229050 0.85 PLAU (0.56) PLAUCCR1CCR5CCR8ATP4A
Hydrochloric Acid SCHEMBL7240496 0.84 ALDH1A1 (0.47) PLAUCCR1CCR5CCR8MAPT
Hydrochloric Acid SCHEMBL7236046 0.84 PLAU (0.55) PLAUCCR1CCR5CCR8ATP4A
SCHEMBL7231676 0.78 CCR1 (0.56) PLAUCCR1CCR5CCR8MAPT
SCHEMBL7232327 0.78 CCR1 (0.38) PLAUCCR1CCR5CCR8
Hydrochloric Acid SCHEMBL7229297 0.75 TAAR1 (0.62) PLAUCCR1CCR5CCR8ATP4A
SCHEMBL7231484 0.75 CCR1 (0.45) PLAUCCR1CCR5CCR8MAPT
SCHEMBL7834251 0.75 CCR1 (0.45) PLAUCCR1CCR5CCR8MAPT
Hydrochloric Acid SCHEMBL7239801 0.74 CCR1 (0.44) PLAUCCR1CCR5CCR8MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed