SCHEMBL7835362

SCHEMBL7835362

Cn1c(CCCOc2ccc(CC3SC(=O)NC3=O)cc2)nc2cccnc21

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 15/20 0.61
FFAR1 O14842 6/20 0.55
PPARA Q07869 4/20 0.55
HRH3 Q9Y5N1 1/20 0.52
RXRA P19793 2/20 0.49
CYP3A4 P08684 1/20 0.49
ESRRA P11474 1/20 0.48
RARG P13631 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7831811 0.95 PPARG (0.61) PPARGFFAR1PPARAHRH3RXRA
SCHEMBL6903005 0.91 PPARG (0.73) PPARGFFAR1PPARAHRH3ESRRA
SCHEMBL7836370 0.81 FFAR1 (0.65) PPARGFFAR1PPARACYP3A4ESRRA
SCHEMBL7833460 0.80 PPARG (0.42) PPARGFFAR1PPARARXRARARG
SCHEMBL7837758 0.79 PPARG (0.65) PPARGFFAR1PPARARXRAESRRA
SCHEMBL7835674 0.78 FFAR1 (0.69) PPARGFFAR1PPARAESRRA
SCHEMBL6900078 0.77 PPARG (0.69) PPARGFFAR1PPARAHRH3RXRA
SCHEMBL7823495 0.77 PPARG (0.58) PPARGFFAR1PPARAHRH3ESRRA
SCHEMBL7835250 0.77 PPARG (0.73) PPARGFFAR1PPARAHRH3RXRA
SCHEMBL1130955 0.77 PPARG (0.79) PPARGFFAR1PPARAESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676398-B1 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO CO (JP) 2001-10-24 EP disclosed
US-6117893-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 2000-09-12 US disclosed
EP-1022274-A1 Oxazolidinedione and Thiazolidinedione derivatves, their preparation and their use Sankyo Company Limited (JP) 2000-07-26 EP disclosed
US-5977365-A HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
US-5624935-A ANTIDIABETIC AGENTS, HYPOGLYCEMIC AGENTS OR ANTILIPEMIC AGENTS SANKYO COMPANY, LIMITED 1997-04-29 US disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed