SCHEMBL7835543

SCHEMBL7835543

CN(C)C(=S)C(C1CCNCC1)N1CCC(NC(=O)c2cc(Cl)c(N)c3c2OC(C)(C)C3)CC1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 13/20 0.42
HTR1A P08908 1/20 0.42
ADRA2C P18825 1/20 0.42
ACHE P22303 1/20 0.42
PTGS1 P23219 1/20 0.42
ADRA1A P35348 1/20 0.42
HTR3A P46098 1/20 0.42
KCNH2 Q12809 1/20 0.42
PTGES O14684 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584843 0.87 HTR4 (0.55) HTR4HTR1AADRA2CACHEPTGS1
SCHEMBL6586787 0.83 HTR4 (0.41) HTR4HTR1AADRA2CACHEPTGS1
SCHEMBL6586073 0.80 HTR4 (0.56) HTR4HTR1AADRA2CACHEPTGS1
SCHEMBL6586000 0.79 HTR4 (0.51) HTR4HTR1AADRA2CACHEPTGS1
SCHEMBL6586562 0.79 HTR4 (0.67) HTR4ADRA2CACHEADRA1AHTR3A
SCHEMBL6590535 0.76 HTR4 (0.47) HTR4HTR1AADRA2CACHEPTGS1
SCHEMBL8504214 0.75 HTR4 (0.57) HTR4HTR1AADRA2CACHEPTGS1
SCHEMBL6583036 0.75 HTR4 (0.56) HTR4HTR1AADRA2CACHEPTGS1
Fumaric Acid SCHEMBL6588715 0.74 HTR4 (0.55) HTR4HTR1AADRA2CACHEPTGS1
SCHEMBL8503793 0.74 HTR4 (0.60) HTR4HTR1AADRA2CACHEPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076055-A1 1- (1-SUBSTITUTED-4-PIPERIDINYL)METHYL]-4-PIPERIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME AND INTERMEDIATES OF THESE COMPOUNDS Dainippon Pharmaceutical Co., Ltd. (JP) 2001-02-14 EP disclosed