SCHEMBL7836655

SCHEMBL7836655

CC(C)(CNc1ccnc2cc(Cl)ccc12)NCc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.48
CYP1A2 P05177 2/20 0.48
CCR1 P32246 1/20 0.46
CYP2C8 P10632 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
SLC2A1 P11166 1/20 0.45
FERMT2 Q96AC1 3/20 0.45
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833242 0.89 CYP1A2 (0.53) PKMCYP1A2CCR1CYP2C8CYP2D6
Hydrochloric Acid SCHEMBL7826427 0.87 CYP1A2 (0.51) PKMCYP1A2CCR1CYP2C8CYP2D6
SCHEMBL7835244 0.87 CYP1A2 (0.53) PKMCYP1A2CCR1CYP2C8CYP2D6
SCHEMBL7826368 0.87 PKM (0.54) PKMCYP1A2CCR1CYP2C8CYP2D6
Hydrochloric Acid SCHEMBL7838222 0.85 PKM (0.59) PKMCYP1A2CCR1CYP2C8CYP2D6
SCHEMBL7836465 0.85 CYP1A2 (0.51) PKMCYP1A2CCR1CYP2C8CYP2D6
SCHEMBL7835537 0.84 PKM (0.54) PKMCYP1A2CCR1CYP2C8CYP2D6
SCHEMBL4281724 0.83 PKM (0.60) PKMCYP1A2CCR1CYP2C8CYP2D6
Hydrochloric Acid SCHEMBL7840186 0.82 CYP1A2 (0.55) PKMCYP1A2CCR1CYP2C8CYP2D6
SCHEMBL4288006 0.82 PKM (0.72) PKMCYP1A2CCR1CYP2C8CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876346-B1 ANTIMALARIAL QUINOLIN DERIVATIVES HOFFMANN LA ROCHE (CH) 2001-07-25 EP disclosed