SCHEMBL7836742

SCHEMBL7836742

CC(C)C[C@@H](C(=O)NN1CC(=O)NC1=O)[C@H](C/C=C/c1ccccc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 2/20 0.48
GRIK1 P39086 2/20 0.37
GRIK2 Q13002 2/20 0.37
MMP2 P08253 5/20 0.35
MMP3 P08254 5/20 0.35
MMP7 P09237 4/20 0.35
GAA P10253 1/20 0.35
MMP1 P03956 4/20 0.35
MMP8 P22894 2/20 0.35
MMP9 P14780 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35
MMP14 P50281 1/20 0.35
CASP1 P29466 1/20 0.35
CASP3 P42574 1/20 0.35
CASP7 P55210 1/20 0.35
CASP6 P55212 1/20 0.35
CASP8 Q14790 1/20 0.35
HTR2A P28223 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835742 1.00 ADAM17 (0.48) ADAM17GRIK1GRIK2MMP2MMP3
SCHEMBL7955135 0.94 ADAM17 (0.55) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL1844380 0.94 ADAM17 (0.55) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL1844385 0.94 ADAM17 (0.55) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL7955133 0.94 ADAM17 (0.55) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL13274078 0.94 ADAM17 (0.55) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL7960536 0.88 ADAM17 (0.43) ADAM17MMP2MMP3MMP7GAA
SCHEMBL7837197 0.88 ADAM17 (0.43) ADAM17MMP2MMP3MMP7GAA
SCHEMBL7837198 0.88 ADAM17 (0.43) ADAM17MMP2MMP3MMP7GAA
SCHEMBL7827360 0.88 ADAM17 (0.43) ADAM17MMP2MMP3MMP7GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137640-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-10-04 EP disclosed
WO-2000035885-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-22 WO disclosed