SCHEMBL7837743

SCHEMBL7837743

CCCCOC(=O)c1cccc2[nH]c(Cl)nc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.55
TDP1 Q9NUW8 2/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
RIPK1 Q13546 1/20 0.53
ALDH1A1 P00352 10/20 0.50
KDM4E B2RXH2 4/20 0.50
MAPK1 P28482 3/20 0.50
CYP3A4 P08684 3/20 0.50
TP53 P04637 1/20 0.50
LMNA P02545 2/20 0.49
HSD17B10 Q99714 2/20 0.49
POLB P06746 1/20 0.44
CYP1A2 P05177 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MMP1 P03956 1/20 0.43
MMP9 P14780 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4713439 0.85 TSHR (0.52) TSHRTDP1L3MBTL1RIPK1ALDH1A1
SCHEMBL5970048 0.82 DHODH (0.58) TSHRTDP1L3MBTL1RIPK1ALDH1A1
SCHEMBL7837745 0.80 TSHR (0.55) TSHRTDP1L3MBTL1ALDH1A1KDM4E
SCHEMBL2830150 0.80 PKN1 (0.61) RIPK1KDM4EKMT2APARP1PKN1
SCHEMBL11789726 0.77 TSHR (0.57) TSHRTDP1L3MBTL1ALDH1A1KDM4E
SCHEMBL716141 0.77 TSHR (0.57) TSHRTDP1L3MBTL1RIPK1ALDH1A1
SCHEMBL27775909 0.77 TSHR (0.57) TSHRTDP1L3MBTL1ALDH1A1KDM4E
SCHEMBL20449581 0.73 KDM4E (0.60) KDM4EHPGDPARP1
SCHEMBL6170661 0.73 PARP1 (0.64) TSHRRIPK1ALDH1A1KDM4ELMNA
Dibutyl Phthalate SCHEMBL4596231 0.73 TSHR (1.00) TSHRTDP1L3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089993-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2001-04-11 EP disclosed
WO-2000000487-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2000-01-06 WO disclosed