SCHEMBL7840650

SCHEMBL7840650

O=C(CCCl)N1Cc2ccccc2Oc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGER2 P43116 1/20 0.50
MAPT P10636 2/20 0.48
TP53 P04637 2/20 0.48
PTGER1 P34995 1/20 0.47
LMNA P02545 2/20 0.46
HSD17B3 P37058 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
ALOX15 P16050 1/20 0.46
CYP2C19 P33261 1/20 0.46
THPO P40225 1/20 0.46
PMP22 Q01453 1/20 0.46
KMT2A Q03164 1/20 0.46
TSHR P16473 1/20 0.43
P2RX4 Q99571 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1366112 0.84 HSD17B3 (0.49) PTGER2MAPTTP53PTGER1LMNA
SCHEMBL1366120 0.80 HDAC3 (0.53) PTGER2MAPTTP53PTGER1LMNA
SCHEMBL7837075 0.80 TSHR (0.51) MAPTTP53HSD17B3MEN1ALDH1A1
SCHEMBL6988456 0.79 HSD17B3 (0.69) MAPTHSD17B3MEN1ALDH1A1CYP1A2
SCHEMBL8788236 0.79 HSD17B3 (0.53) PTGER2MAPTHSD17B3MEN1ALDH1A1
SCHEMBL11545122 0.74 MEN1 (0.53) PTGER2MAPTPTGER1HSD17B3MEN1
SCHEMBL9185113 0.73 MAPT (0.64) PTGER2MAPTTP53PTGER1HSD17B3
SCHEMBL4637311 0.72 TSHR (0.81) MAPTTP53MEN1ALDH1A1KMT2A
SCHEMBL7344478 0.71 P2RX4 (0.54) MAPTHSD17B3MEN1ALDH1A1CYP1A2
SCHEMBL1367874 0.70 NPC1 (0.47) MAPTTP53LMNAMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820450-B1 N-substituted azaheterocyclic carboxylic acids and alkylesters thereof NOVO NORDISK AS (DK) 2001-09-12 EP disclosed
EP-0820450-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1998-01-28 EP disclosed
WO-1996031497-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed