SCHEMBL7837075

SCHEMBL7837075

O=C(CCCl)N1Cc2ccccc2Cc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.51
MAPT P10636 3/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
HSD17B3 P37058 3/20 0.47
NOTUM Q6P988 4/20 0.47
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MITF O75030 1/20 0.44
ALDH1A1 P00352 2/20 0.43
POLB P06746 1/20 0.43
TP53 P04637 1/20 0.43
NFKB1 P19838 1/20 0.43
MAPK1 P28482 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CASP3 P42574 1/20 0.41
CASP2 P42575 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7840650 0.80 PTGER2 (0.50) TSHRMAPTKMT2AMEN1HSD17B3
SCHEMBL4637311 0.79 TSHR (0.81) TSHRMAPTKMT2AMEN1NOTUM
SCHEMBL3270957 0.79 ALDH1A1 (0.46) TSHRMAPTKMT2AMEN1HSD17B3
SCHEMBL5251752 0.77 TSHR (0.67) TSHRMAPTKMT2AMEN1NOTUM
SCHEMBL24817140 0.76 NOTUM (0.52) TSHRMAPTKMT2AMEN1NOTUM
SCHEMBL29987139 0.76 NOTUM (0.52) TSHRMAPTKMT2AMEN1NOTUM
SCHEMBL19404981 0.75 HSD17B3 (0.64) TSHRMAPTKMT2AMEN1HSD17B3
SCHEMBL24201501 0.74 HSD17B3 (0.67) TSHRMAPTKMT2AMEN1HSD17B3
SCHEMBL8558342 0.73 HPGD (0.48) KMT2AHSD17B3NPC1RAB9AALDH1A1
SCHEMBL19014017 0.73 HSD17B3 (0.60) TSHRMAPTKMT2AMEN1HSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820450-B1 N-substituted azaheterocyclic carboxylic acids and alkylesters thereof NOVO NORDISK AS (DK) 2001-09-12 EP disclosed
EP-0820450-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1998-01-28 EP disclosed
WO-1996031497-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed