SCHEMBL7841197

SCHEMBL7841197

CCCCOC(=O)NN1CCC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
NPC1 O15118 2/20 0.47
MAPT P10636 2/20 0.47
RAB9A P51151 2/20 0.47
TP53 P04637 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
KMT2A Q03164 1/20 0.47
RELA Q04206 1/20 0.47
EPHX1 P07099 1/20 0.46
ACHE P22303 11/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1383077 0.96 SMN1; SMN2 (0.50) SMN1; SMN2NPC1MAPTRAB9ATP53
SCHEMBL3010245 0.95 SMN1; SMN2 (0.52) SMN1; SMN2NPC1MAPTRAB9ATP53
SCHEMBL8589909 0.90 EPHX1 (0.56) SMN1; SMN2NPC1MAPTRAB9ATP53
SCHEMBL8590406 0.88 EPHX1 (0.54) SMN1; SMN2NPC1MAPTRAB9ATP53
SCHEMBL7194159 0.86 EPHX1 (0.59) SMN1; SMN2EPHX1ACHEGAA
SCHEMBL28783627 0.85 GNAI3 (0.55) SMN1; SMN2NPC1MAPTRAB9ATP53
SCHEMBL6381523 0.83 SMN1; SMN2 (0.40) SMN1; SMN2NPC1MAPTRAB9ATP53
SCHEMBL7009651 0.82 EPHX1 (0.40) SMN1; SMN2NPC1MAPTRAB9ATP53
SCHEMBL6582896 0.82 MAPT (0.47) SMN1; SMN2NPC1MAPTRAB9ATP53
SCHEMBL5747211 0.82 SMN1; SMN2 (0.40) SMN1; SMN2NPC1MAPTRAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102762-A2 2-SUBSTITUTED-1-PIPERIDYL BENZIMIDAZOLE COMPOUNDS AS ORL1-RECEPTOR AGONISTS PFIZER INC. (US) 2001-05-30 EP disclosed
WO-2000008013-A2 2-SUBSTITUTED-1-PIPERIDYL BENZIMIDAZOLE COMPOUNDS AS ORL1-RECEPTOR AGONISTS PFIZER PHARMACEUTICALS INC. (JP) 2000-02-17 WO disclosed