SCHEMBL7841929

SCHEMBL7841929

CCOC(=O)c1cn2cccc(OCCCCN3C(=O)CSC3=O)c2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 3/20 0.43
HPGD P15428 2/20 0.43
GAA P10253 2/20 0.43
HSD17B10 Q99714 1/20 0.43
NPSR1 Q6W5P4 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 2/20 0.38
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
HTT P42858 1/20 0.36
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
DRD4 P21917 1/20 0.34
HTR2A P28223 1/20 0.34
DRD3 P35462 1/20 0.34
TBXAS1 P24557 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7845274 0.85 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDGAAHSD17B10
SCHEMBL10646314 0.81 KDM4E (0.53) ALDH1A1KDM4EHPGDGAAMEN1
SCHEMBL7836177 0.80 KDM4E (0.39) ALDH1A1KDM4EHPGDGAAMEN1
SCHEMBL7836178 0.80 KDM4E (0.39) ALDH1A1KDM4EHPGDGAAMEN1
Hydrochloric Acid SCHEMBL7844019 0.79 KDM4E (0.38) ALDH1A1KDM4EHPGDGAAMEN1
Hydrochloric Acid SCHEMBL7841644 0.79 KDM4E (0.38) ALDH1A1KDM4EHPGDGAAMEN1
SCHEMBL7835071 0.79 HRH3 (0.42) ALDH1A1KDM4EHPGDHSD17B10NPSR1
SCHEMBL7842563 0.77 ALDH1A1 (0.42) ALDH1A1KDM4EGAAHSD17B10MEN1
SCHEMBL1202722 0.74 KDM4E (0.55) ALDH1A1KDM4EHPGDGAAHSD17B10
SCHEMBL7844901 0.73 ALDH1A1 (0.43) ALDH1A1KDM4EGAAHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767790-B1 CONDENSED IMIDAZOLE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-12-12 EP disclosed
US-5840732-A ANTIDIABETIC AGENTS, AUTOIMMUNE DISEASES OR IMMUNOSUPPRESSANTS TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 1998-11-24 US disclosed
EP-0767790-A1 CONDENSED IMIDAZOLE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-04-16 EP disclosed
WO-1995035296-A1 CONDENSED IMIDAZOLE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-28 WO disclosed