SCHEMBL78424

SCHEMBL78424

COCCOCc1cc(OC)cc(C(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.36
CALM1 P0DP23 2/20 0.35
MAPT P10636 1/20 0.34
PTGS2 P35354 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
EPHX2 P34913 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
HMGCR P04035 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4602449 0.78 TACR1 (0.52) TACR1CALM1ALDH1A1
SCHEMBL14838199 0.78 TACR1 (0.38) TACR1GABRA1GABRB2L3MBTL1HMGCR
SCHEMBL88992 0.78 PTGS2 (0.37) TACR1CALM1PTGS2GABRA1GABRG2
SCHEMBL4602443 0.77 TACR1 (0.35) TACR1CALM1PTGS2GABRA1GABRG2
SCHEMBL90337 0.77 DAO (0.41) TACR1CALM1MAPTPTGS2GABRA1
SCHEMBL8265190 0.77 TACR1 (0.35) TACR1CALM1PTGS2GABRA1GABRG2
SCHEMBL8264225 0.77 TACR1 (0.35) TACR1CALM1PTGS2GABRA1GABRG2
SCHEMBL1204935 0.76 NR1H4 (0.38) TACR1MAPTL3MBTL1MEN1NPC1
SCHEMBL22861019 0.75 PTGS2 (0.41) CALM1PTGS2GABRA1GABRG2GABRB3
SCHEMBL1205032 0.75 CA1 (0.43) MAPTCA1CA2L3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed