SCHEMBL7842726

SCHEMBL7842726

NS(=O)(=O)c1ccc(-c2sc(-c3ccc(Cl)cc3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.78
PTGS1 P23219 6/20 0.71
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15689086 0.89 PTGS2 (0.67) PTGS2PTGS1CA12CA1CA2
SCHEMBL7845380 0.89 PTGS2 (0.77) PTGS2PTGS1
SCHEMBL7845406 0.88 PTGS2 (0.69) PTGS2PTGS1
SCHEMBL7844918 0.88 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL7840831 0.88 PTGS2 (0.78) PTGS2PTGS1
SCHEMBL15688673 0.88 PTGS2 (0.65) PTGS2PTGS1CA12CA1CA2
SCHEMBL15688973 0.86 PTGS2 (0.61) PTGS2PTGS1CA12CA1CA2
SCHEMBL7843422 0.85 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL7845580 0.85 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL7845977 0.85 PTGS2 (0.80) PTGS2PTGS1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1125932-A2 Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 2001-08-22 EP disclosed
US-5668161-A Substituted thiazoles for the treatment of inflammation G.D. SEARLE & CO. (US) 1997-09-16 US disclosed
EP-0772606-A1 SUBSTITUTED THIAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-05-14 EP disclosed
WO-1996003392-A1 SUBSTITUTED THIAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed