SCHEMBL7843018

SCHEMBL7843018

O=C(c1c[nH]c2ccc(C=CCO)cc2c1=O)N(CCN1CCOCC1)Cc1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.42
HPGD P15428 6/20 0.42
KDM4E B2RXH2 5/20 0.42
GAA P10253 3/20 0.42
GLA P06280 1/20 0.42
MAPT P10636 2/20 0.40
TSHR P16473 3/20 0.40
HSD17B10 Q99714 2/20 0.40
TACR2 P21452 1/20 0.39
CFTR P13569 1/20 0.38
USP2 O75604 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPK1 P28482 2/20 0.38
LMNA P02545 2/20 0.38
THRB P10828 1/20 0.38
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 2/20 0.37
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6668634 0.79 TP53 (0.46) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL7841900 0.79 TP53 (0.46) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL6670162 0.79 HTR2A (0.43) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL7846819 0.78 HTR2A (0.43) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL6701498 0.77 ALDH1A1 (0.43) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL6667851 0.76 ALDH1A1 (0.42) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL6667925 0.76 ALDH1A1 (0.45) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL6667863 0.76 ALDH1A1 (0.43) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL7848149 0.75 POLB (0.42) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL7845988 0.75 ALDH1A1 (0.43) ALDH1A1HPGDKDM4EGAAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140850-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2001-10-10 EP claimed
WO-2000040561-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2000-07-13 WO claimed
EP-1140850-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2001-10-10 EP disclosed
WO-2000040561-A1 QUINOLINECARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2000-07-13 WO disclosed