SCHEMBL7843430

SCHEMBL7843430

COc1ccc(/C=C2/C(=O)Nc3ccccc32)cc1OC

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.76
DHFR P00374 1/20 0.74
PDE4A P27815 2/20 0.67
PDE4B Q07343 2/20 0.67
PDE4C Q08493 2/20 0.67
PDE4D Q08499 2/20 0.67
PDE3B Q13370 1/20 0.67
PDE3A Q14432 1/20 0.67
NPC1 O15118 1/20 0.65
CSNK1D P48730 3/20 0.64
CSNK1A1 P48729 2/20 0.64
CSNK1E P49674 2/20 0.64
L3MBTL1 Q9Y468 1/20 0.64
GMNN O75496 1/20 0.64
ALDH1A1 P00352 1/20 0.64
LMNA P02545 1/20 0.64
TP53 P04637 1/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
MAPT P10636 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5477780 1.00 ERBB2 (0.76) ERBB2DHFRPDE4APDE4BPDE4C
SCHEMBL5477779 1.00 ERBB2 (0.76) ERBB2DHFRPDE4APDE4BPDE4C
SCHEMBL5595791 0.90 ERBB2 (0.72) ERBB2DHFRPDE4APDE4BPDE4C
SCHEMBL3374408 0.90 ERBB2 (0.72) ERBB2DHFRPDE4APDE4BPDE4C
SCHEMBL6405474 0.88 ERBB2 (0.71) ERBB2DHFRPDE4APDE4BPDE4C
SCHEMBL5476202 0.88 DHFR (0.73) ERBB2DHFRPDE4APDE4BPDE4C
SCHEMBL5476200 0.88 DHFR (0.73) ERBB2DHFRPDE4APDE4BPDE4C
SCHEMBL5469649 0.88 DHFR (0.77) ERBB2DHFRNPC1CSNK1DCSNK1A1
SCHEMBL6405476 0.88 ERBB2 (0.71) ERBB2DHFRPDE4APDE4BPDE4C
SCHEMBL14448907 0.88 DHFR (0.77) ERBB2DHFRNPC1CSNK1DCSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730579-B1 SUBSTITUTED INDOLES AS PHOSPHODIESTERASE TYPE IV INHIBITORS PFIZER (US) 2001-03-07 EP disclosed