SCHEMBL7844449

SCHEMBL7844449

[CH2]C(c1ncc(-c2ncc[nH]2)c(-c2ccc(Cl)cc2Cl)n1)N(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.44
CCNB2 O95067 2/20 0.43
CDK1 P06493 2/20 0.43
CCNB1 P14635 2/20 0.43
GSK3A P49840 2/20 0.43
CCNB3 Q8WWL7 2/20 0.43
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ROS1 P08922 1/20 0.35
CRHR1 P34998 7/20 0.34
CNR1 P21554 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MCOLN3 Q8TDD5 1/20 0.34
RPS6KB1 P23443 1/20 0.33
CDK2 P24941 1/20 0.33
LIMK1 P53667 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4393755 0.79 GSK3B (0.50) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL4393758 0.79 ROS1 (0.53) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL5093917 0.78 GSK3B (0.47) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL4398386 0.78 GSK3B (0.41) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL7024110 0.77 GSK3B (0.44) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL4972846 0.77 GSK3B (0.52) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL7022602 0.76 GSK3B (0.63) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL5089268 0.76 GSK3B (0.48) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL27538055 0.76 GSK3B (0.57) GSK3BCCNB2CDK1CCNB1GSK3A
SCHEMBL5099514 0.76 GSK3B (0.46) GSK3BCCNB2CDK1CCNB1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed