SCHEMBL7844941

SCHEMBL7844941

COc1ccnc(-c2ccccc2N)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.61
CCR5 P51681 1/20 0.61
CCR8 P51685 1/20 0.61
NOS3 P29474 2/20 0.53
NOS1 P29475 2/20 0.53
NOS2 P35228 2/20 0.53
ADORA3 P0DMS8 1/20 0.47
PLAU P00749 1/20 0.45
NPC1 O15118 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
HSD17B10 Q99714 1/20 0.42
RAB9A P51151 1/20 0.42
SCN2A Q99250 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231911 0.81 CCR1 (0.63) CCR1CCR5CCR8NOS3NOS1
SCHEMBL27909626 0.80 CCR1 (0.61) CCR1CCR5CCR8NOS3NOS1
SCHEMBL29395249 0.78 CCR1 (1.00) CCR1CCR5CCR8NOS3NOS1
SCHEMBL182529 0.78 CCR1 (1.00) CCR1CCR5CCR8NOS3NOS1
SCHEMBL25192476 0.78 CCR1 (0.58) CCR1CCR5CCR8NOS3NOS1
SCHEMBL10333208 0.78 CCR1 (0.58) CCR1CCR5CCR8NOS3NOS1
SCHEMBL27927335 0.78 CCR1 (0.58) CCR1CCR5CCR8NOS3NOS1
SCHEMBL7230635 0.76 CCR1 (0.56) CCR1CCR5CCR8NOS3NOS1
SCHEMBL8746042 0.76 CCR1 (0.95) CCR1CCR5CCR8NOS3NOS1
Methane SCHEMBL21386924 0.76 CCR1 (0.95) CCR1CCR5CCR8NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed