SCHEMBL7845153

SCHEMBL7845153

O=C1Cc2ccccc2N1c1ccc(Br)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.53
MEN1 O00255 4/20 0.53
CASP6 P55212 4/20 0.53
GAA P10253 3/20 0.53
HPGD P15428 1/20 0.53
MAPT P10636 2/20 0.46
ALOX12 P18054 2/20 0.46
ALOX15 P16050 1/20 0.43
HBB P68871 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CASP3 P42574 2/20 0.42
SENP8 Q96LD8 2/20 0.42
SENP7 Q9BQF6 2/20 0.42
SENP6 Q9GZR1 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
GRM1 Q13255 3/20 0.41
NOTUM Q6P988 1/20 0.40
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
PMP22 Q01453 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11133610 0.84 HPGD (0.62) KMT2AMEN1CASP6GAAHPGD
SCHEMBL6328308 0.78 HPGD (0.74) KMT2AMEN1CASP6GAAHPGD
SCHEMBL6772536 0.77 HPGD (0.68) KMT2AMEN1CASP6GAAHPGD
SCHEMBL7845228 0.76 HPGD (0.57) KMT2AMEN1CASP6GAAHPGD
SCHEMBL3027278 0.75 CYP3A4 (0.50) KMT2AMEN1CASP6GAAHPGD
SCHEMBL29651988 0.74 GAA (0.59) KMT2AMEN1CASP6GAAHPGD
SCHEMBL2982634 0.74 GAA (0.59) KMT2AMEN1CASP6GAAHPGD
SCHEMBL4692980 0.74 HPGD (0.69) KMT2AMEN1CASP6GAAHPGD
SCHEMBL11563108 0.74 HPGD (0.54) KMT2AMEN1CASP6GAAHPGD
SCHEMBL10562313 0.73 KMT2A (0.77) KMT2AMEN1CASP6GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105376-A1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2001-06-13 EP disclosed
WO-2000010975-A1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 2000-03-02 WO disclosed