SCHEMBL7845547

SCHEMBL7845547

COC(=O)c1ccc(NC2CCCCC2)c(C#Cc2ccc(OCc3cc(OC)ccc3-c3ccc(Cl)cc3)cc2)c1.COC(=O)c1ccc2c(c1)cc(-c1ccc(OCc3cc(OC)ccc3-c3ccc(Cl)cc3)cc1)n2C1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.36
PTGS2 P35354 4/20 0.33
TACR2 P21452 1/20 0.33
TACR1 P25103 1/20 0.33
MAPK10 P53779 3/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
ALDH1A1 P00352 1/20 0.31
ATM Q13315 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HPGD P15428 1/20 0.31
CNR1 P21554 1/20 0.31
VDR P11473 2/20 0.31
POLB P06746 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE7A Q13946 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5524346 0.90 TACR2 (0.39) NR1H4PTGS2TACR2TACR1HTT
SCHEMBL5514514 0.89 PTGS2 (0.38) NR1H4PTGS2TACR2TACR1SMN1; SMN2
SCHEMBL791555 0.83 NR1H4 (0.41) NR1H4PTGS2VDR
SCHEMBL5519425 0.80 TACR2 (0.38) NR1H4TACR2TACR1SMN1; SMN2HPGD
SCHEMBL5514105 0.79 NR1H4 (0.47) NR1H4PTGS2CNR1VDR
SCHEMBL5508934 0.74 MAPT (0.47) NR1H4ALDH1A1NPSR1VDR
SCHEMBL5527483 0.73 NR1H4 (0.51) NR1H4VDR
Hydrochloric Acid SCHEMBL5512953 0.73 NR1H4 (0.49) NR1H4VDR
Hydrochloric Acid SCHEMBL5515106 0.72 NR1H4 (0.50) NR1H4VDR
SCHEMBL5509930 0.72 RPS6KB1 (0.45) NR1H4CNR1VDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1162196-A1 FUSED-RING COMPOUNDS AND USE THEREOF AS DRUGS JAPAN TOBACCO INC. (JP) 2001-12-12 EP disclosed