SCHEMBL7846039

SCHEMBL7846039

CC(C)(C)OC(=O)NC(N)=Nc1cccc(-c2ncccc2CO[Si](C)(C)C(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 8/20 0.36
ITGB3 P05106 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGAV P06756 1/20 0.35
ITGA2B P08514 1/20 0.35
ITGB5 P18084 1/20 0.35
HRH4 Q9H3N8 8/20 0.35
HRH3 Q9Y5N1 5/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
HRH1 P35367 4/20 0.34
BACE1 P56817 1/20 0.33
NQO2 P16083 1/20 0.32
KDM4E B2RXH2 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NPFFR1 Q9GZQ6 1/20 0.32
NPFFR2 Q9Y5X5 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
GABRA5 P31644 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7237052 0.92 NPFFR1 (0.37) ITGB3ITGB1ITGAVITGA2BITGB5
SCHEMBL7847203 0.85 BACE1 (0.32) ITGB3ITGB1ITGAVITGA2BITGB5
SCHEMBL7843840 0.85 HRH2 (0.34) HRH2ITGB3ITGB1ITGAVITGA2B
SCHEMBL7846042 0.79 CYP17A1 (0.34) BACE1KDM4EALDH1A1MAPT
SCHEMBL7847206 0.78 NQO2 (0.34) BACE1NQO2KDM4EL3MBTL1ACACB
SCHEMBL7236713 0.76 NPFFR1 (0.35) ITGB3ITGB1ITGAVITGA2BITGB5
SCHEMBL7846035 0.76 ITGB3 (0.34) HRH2ITGB3ITGB1ITGAVITGA2B
SCHEMBL7846044 0.76 ITGB3 (0.34) HRH2ITGB3ITGB1ITGAVITGA2B
SCHEMBL7237877 0.74 TRPV1 (0.40) ITGB3ITGB1ITGAVITGA2BITGB5
SCHEMBL7230890 0.73 MAP4K4 (0.40) BACE1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed