SCHEMBL7846259

SCHEMBL7846259

CCCCCCOc1ccc2[nH]c(C)c(CC[C@H](CO[Si](C)(C)C(C)(C)C)n3cnc(C(N)=O)c3)c2c1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADA P00813 15/20 0.55
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
HTR1D P28221 2/20 0.34
HTR1B P28222 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7850071 0.90 ADA (0.56) ADA
SCHEMBL7847452 0.90 ADA (0.67) ADAGABRA1GABRG2GABRB3GABRA5
SCHEMBL7848923 0.86 CYP1A2 (0.41) ADAHTR1D
SCHEMBL6938856 0.83 ADA (0.80) ADA
SCHEMBL7848399 0.81 ADA (0.54) ADAHTR1DHTR1B
SCHEMBL7836767 0.79 ADA (0.68) ADA
SCHEMBL6936319 0.77 ADA (0.80) ADA
SCHEMBL6941256 0.77 ADA (0.80) ADA
SCHEMBL7846263 0.77 ADA (0.48) ADAHTR1DHTR1B
SCHEMBL6938448 0.75 ADA (0.79) ADA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161429-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed
WO-2000055155-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-21 WO disclosed