SCHEMBL7846263

SCHEMBL7846263

CCCCCCOCc1ccc2[nH]cc(CC[C@H](CO[Si](C)(C)C(C)(C)C)n3cnc(C(N)=O)c3)c2c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADA P00813 9/20 0.48
HTR1B P28222 9/20 0.37
HTR1A P08908 8/20 0.37
HTR1D P28221 8/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
KDM4E B2RXH2 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
HTR2A P28223 1/20 0.37
CYP2C19 P33261 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7848925 0.87 ADA (0.44) ADA
SCHEMBL7847893 0.85 ADA (0.43) ADAHTR1BHTR1AHTR1DMAPT
SCHEMBL7848399 0.84 ADA (0.54) ADAHTR1BHTR1AHTR1DMAPT
SCHEMBL7836809 0.81 ADA (0.43) ADAHTR2A
SCHEMBL7850190 0.79 ADA (0.43) ADACYP2C19
SCHEMBL7847420 0.78 ADA (0.49) ADAHTR1DMAPTKDM4EMEN1
SCHEMBL7846259 0.77 ADA (0.55) ADAHTR1BHTR1D
SCHEMBL6938856 0.77 ADA (0.80) ADA
SCHEMBL7850266 0.76 PTPRA (0.41) ADAHTR1AHTR1DMAPTCYP2C19
SCHEMBL7847454 0.75 ADA (0.41) ADAHTR1BHTR1AHTR1DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161429-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed
WO-2000055155-A2 HETEROCYCLIC COMPOUNDS AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-21 WO disclosed