SCHEMBL7846656

SCHEMBL7846656

COC(=O)c1cccnc1-c1cccc(/N=C(\N)N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.38
METAP2 P50579 1/20 0.35
FAAH O00519 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
RORB Q92753 1/20 0.33
LHCGR P22888 1/20 0.33
ATR Q13535 1/20 0.33
CFTR P13569 1/20 0.32
SLC40A1 Q9NP59 1/20 0.32
F2 P00734 2/20 0.32
F10 P00742 2/20 0.32
PRSS1 P07477 2/20 0.32
PRSS2 P07478 2/20 0.32
PRSS3 P35030 2/20 0.32
MAP2K1 Q02750 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846658 1.00 ALOX5AP (0.38) ALOX5APMETAP2FAAHTDP1RORB
SCHEMBL7240056 0.90 KDM4E (0.39) TDP1RORBF2F10PRSS1
SCHEMBL7240054 0.90 KDM4E (0.39) TDP1RORBF2F10PRSS1
SCHEMBL7842304 0.86 TRPV1 (0.37) LHCGR
SCHEMBL7846907 0.86 TRPV1 (0.35)
SCHEMBL7842303 0.86 TRPV1 (0.37) LHCGR
SCHEMBL7232510 0.82 ATR (0.39) ALOX5APMETAP2FAAHTDP1RORB
SCHEMBL7845852 0.82 TRPV1 (0.41) TDP1NPC1RAB9ASMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL7232462 0.81 TAAR1 (0.44) ALOX5APMETAP2TDP1RORBPRSS1
SCHEMBL7847203 0.80 BACE1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed