SCHEMBL7846907

SCHEMBL7846907

Cc1cccnc1-c1cccc(N=C(N)N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 9/20 0.35
CYP2A6 P11509 1/20 0.35
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
CETP P11597 1/20 0.33
BACE1 P56817 2/20 0.33
MGLL Q99685 1/20 0.33
CTSD P07339 1/20 0.33
ABL1 P00519 1/20 0.33
PLAU P00749 1/20 0.33
FGFR3 P22607 1/20 0.32
KDR P35968 1/20 0.32
GRIA2 P42262 1/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7842304 0.90 TRPV1 (0.37) TRPV1FGFR3KDR
SCHEMBL7842303 0.90 TRPV1 (0.37) TRPV1FGFR3KDR
SCHEMBL7240054 0.88 KDM4E (0.39)
SCHEMBL7240056 0.88 KDM4E (0.39)
SCHEMBL7846656 0.86 ALOX5AP (0.38)
SCHEMBL7846658 0.86 ALOX5AP (0.38)
SCHEMBL7845852 0.85 TRPV1 (0.41) TRPV1SIGMAR1
SCHEMBL7847203 0.83 BACE1 (0.32) BACE1
SCHEMBL7846734 0.81 CNR1 (0.39) CYP2A6ABL1PLAUFGFR3KDR
SCHEMBL7846731 0.81 CNR1 (0.39) CYP2A6ABL1PLAUFGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed