SCHEMBL7846864

SCHEMBL7846864

NC(=O)C(C(N)=O)(C(=O)c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.50
KMT2A Q03164 1/20 0.50
CES1 P23141 4/20 0.48
TSHR P16473 2/20 0.48
CYP2C19 P33261 2/20 0.48
POLB P06746 1/20 0.48
CYP3A4 P08684 1/20 0.48
PARP1 P09874 1/20 0.48
RECQL P46063 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
KCNN4 O15554 7/20 0.44
HTT P42858 1/20 0.42
CES2 O00748 2/20 0.41
DAO P14920 1/20 0.41
NAPRT Q6XQN6 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1666976 0.87 CES1 (0.61) MAPTKMT2ACES1TSHRCYP2C19
SCHEMBL7039215 0.76 MAPT (0.57) MAPTKMT2ACES1TSHRCYP2C19
SCHEMBL1669227 0.75 CES1 (0.57) MAPTKMT2ACES1POLBCYP3A4
SCHEMBL27914495 0.74 MAPT (0.52) MAPTKMT2ACES1TSHRCYP2C19
SCHEMBL1878464 0.74 CES1 (0.52) MAPTKMT2ACES1TSHRCYP2C19
SCHEMBL1508202 0.73 CES1 (0.56) MAPTCES1TSHRCYP2C19POLB
SCHEMBL15519395 0.73 CES1 (0.56) MAPTCES1TSHRCYP2C19POLB
SCHEMBL461653 0.72 CES1 (0.50) MAPTKMT2ACES1TSHRCYP2C19
SCHEMBL1168769 0.72 CES1 (0.50) MAPTKMT2ACES1TSHRCYP2C19
SCHEMBL8020656 0.72 MAPT (0.52) MAPTKMT2ACES1TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150565-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION bioscience AG (DE) 2001-11-07 EP claimed
WO-2000045635-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2000-08-10 WO claimed