SCHEMBL8020656

SCHEMBL8020656

CC(C)(C(N)=O)C(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
KMT2A Q03164 1/20 0.52
CES1 P23141 5/20 0.50
TSHR P16473 4/20 0.50
HSD17B10 Q99714 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
CYP2C19 P33261 2/20 0.50
POLB P06746 1/20 0.50
CYP3A4 P08684 1/20 0.50
PARP1 P09874 1/20 0.50
RECQL P46063 1/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
SRC P12931 1/20 0.46
ALDH1A1 P00352 4/20 0.42
CES2 O00748 3/20 0.42
DAO P14920 1/20 0.42
NAPRT Q6XQN6 1/20 0.42
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4618681 0.86 CES1 (0.58) MAPTKMT2ACES1TSHRHSD17B10
SCHEMBL8600048 0.83 CES1 (0.47) MAPTKMT2ACES1TSHRHSD17B10
SCHEMBL819138 0.82 CES1 (0.54) MAPTKMT2ACES1TSHRHSD17B10
SCHEMBL27571079 0.81 CA2 (0.50) MAPTKMT2ACES1TDP1ALDH1A1
SCHEMBL12913259 0.80 CES1 (0.52) MAPTCES1TSHRHSD17B10TDP1
SCHEMBL28304793 0.80 CES1 (0.52) MAPTCES1TSHRHSD17B10TDP1
SCHEMBL11011559 0.78 CES1 (0.50) MAPTKMT2ACES1TSHRHSD17B10
SCHEMBL7039215 0.78 MAPT (0.57) MAPTKMT2ACES1TSHRHSD17B10
SCHEMBL28192063 0.77 LMNA (0.61) TDP1POLBCYP3A4L3MBTL1ALDH1A1
SCHEMBL9632467 0.77 CES1 (0.54) MAPTKMT2ACES1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093323-B Beta-functionalized chiral homoallylic alcohol derivative and preparation method and application thereof 武汉大学 2023-12-22 CN disclosed
CN-114057666-B Synthesis method of 4, 5-disubstituted-2-aminothiazole compound 沈阳药科大学 2023-02-07 CN disclosed
CN-115093323-A Beta-functionalized chiral homoallyl alcohol derivative and preparation method and application thereof 武汉大学 2022-09-23 CN disclosed
CN-114989035-A Sulfuryl fluoride promoted reaction method for converting beta-diketone to alkyne 扬州工业职业技术学院 2022-09-02 CN disclosed
CN-114057666-A Synthesis method of 4, 5-disubstituted-2-aminothiazole compound 沈阳药科大学 2022-02-18 CN disclosed
CN-107548397-B Kv1.3 inhibitors and medical uses thereof 4SC股份公司 2020-12-29 CN disclosed
CN-107548396-B Kv1.3 inhibitors and medical uses thereof 4SC股份公司 2020-04-28 CN disclosed
CN-106478443-B The method that difluoro Ya Jia Ji Phosphonium inner salts are used to synthesize β keto-amides as new ammonolysis reagent 四川理工学院 2018-04-03 CN disclosed
CN-107548396-A Kv1.3 inhibitors and medical uses thereof 4SC股份公司 2018-01-05 CN disclosed
CN-107548397-A Kv1.3 inhibitors and medical uses thereof 4SC股份公司 2018-01-05 CN disclosed
CN-106478443-A The method that difluoro methylene inner salt is used for synthesizing β keto-amide as new ammonolysis reagent 四川理工学院 2017-03-08 CN disclosed
CN-102321066-B Method for producing aryl-aminopropanols SALTIGO GMBH 2014-07-23 CN disclosed
CN-1445224-B Process for preparing arylaminopropanols SALTIGO GMBH 2012-07-11 CN disclosed
CN-102321066-A The method for preparing the arylamino propyl alcohol SALTIGO GMBH 2012-01-18 CN disclosed
CN-1445224-A Process for preparing arylaminopropanols BAYER AG (DE) 2003-10-01 CN disclosed
EP-0973856-A1 N-ACYL OXAZIRIDINES AS BLEACH AGENTS UNILEVER N.V. (NL) 2000-01-26 EP disclosed
WO-1998045397-A1 N-ACYL OXAZIRIDINES AS BLEACH AGENTS UNILEVER N.V. (NL) 1998-10-15 WO disclosed
US-5755991-A USEFUL IN CLEANING FABRICS, HOUSEHOLD FIXTURES, TABLEWARE AND DENTURES LEVER BROTHERS COMPANY, DIVISION OF CONOPCO, INC. (US) 1998-05-26 US disclosed