SCHEMBL7847544

SCHEMBL7847544

[CH2]c1cccc(OC)c1N(CC)C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
POLB P06746 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CTSD P07339 1/20 0.36
KMT2A Q03164 2/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
TSHR P16473 1/20 0.36
LMNA P02545 2/20 0.36
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208682 0.80 CA12 (0.41) TP53CA12CA1CA2CA7
SCHEMBL4286533 0.75 ESR1 (0.48) CA12CA1CA2CA7CA9
SCHEMBL23028186 0.73 CA12 (0.43) TP53CA12CA1CA2CA7
SCHEMBL1857458 0.72 CA12 (0.42) CA12CA1CA2CA7CA9
SCHEMBL9021597 0.69 CA12 (0.46) TP53CA12CA1CA2CA7
SCHEMBL11659047 0.68 ATM (0.38) TP53HSD17B10CTSDKMT2AMAPK1
SCHEMBL12427635 0.68 HTT (0.50) TP53CA12CA1CA2CA7
SCHEMBL30705345 0.67 CA12 (0.47) TP53CA12CA1CA2CA7
SCHEMBL11100795 0.67 TP53 (0.53) TP53CA12CA1CA2CA7
SCHEMBL2754166 0.67 ESR1 (0.46) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1121363-A2 6-SUBSTITUTED PYRAZOLO 3,4-d]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS Du Pont Pharmaceuticals Company (US) 2001-08-08 EP claimed
WO-2000021926-A2 6-SUBSTITUTED PYRAZOLO[3,4-d]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 2000-04-20 WO claimed