SCHEMBL6208682

SCHEMBL6208682

[CH2]c1cccc(OC)c1N(C)C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 2/20 0.41
CA4 P22748 1/20 0.38
ALDH1A1 P00352 4/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 2/20 0.36
CTSD P07339 1/20 0.36
HTT P42858 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847544 0.80 TP53 (0.38) CA12CA1CA2CA7CA9
SCHEMBL6210954 0.78 THRB (0.35) CA12CA1CA2CA7CA9
SCHEMBL9021597 0.73 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL24393532 0.70 CA1 (0.47) CA12CA1CA2CA7CA9
SCHEMBL30705345 0.70 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL8516410 0.70 S1PR4 (0.41) CA12CA1CA2CA7CA9
1,2-Dimethoxybenzene SCHEMBL28118612 0.68 CA1 (0.72) CA12CA1CA2CA7CA9
SCHEMBL8483409 0.67 CA12 (0.74) CA12CA1CA2CA7CA9
SCHEMBL9524209 0.67 CA12 (0.47) CA12CA1CA2CA7CA9
Acetic Acid SCHEMBL27619403 0.66 CA1 (0.50) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383769-A4 6-SUBSTITUTED PYRAZOLO 3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2005-08-03 EP disclosed
EP-1383769-A2 6-SUBSTITUTED PYRAZOLO 3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS Bristol-Myers Squibb Pharma Company (US) 2004-01-28 EP disclosed
WO-2002067654-A2 6-SUBSTITUTED PYRAZOLO[3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-09-06 WO disclosed