SCHEMBL7847701

SCHEMBL7847701

O=C(O)c1ccc(Cc2cc(-c3ccc(C(F)(F)F)cc3)[nH]n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 2/20 0.56
MAPK1 P28482 2/20 0.50
MAP2K4 P45985 2/20 0.50
MAPK6 Q16659 2/20 0.50
MAPKAPK3 Q16644 1/20 0.50
MAPKAPK5 Q8IW41 1/20 0.50
CYP2C8 P10632 1/20 0.46
RXRA P19793 2/20 0.46
RXRB P28702 2/20 0.46
RXRG P48443 2/20 0.46
PPARA Q07869 2/20 0.45
MAP4K4 O95819 1/20 0.44
CSNK2A2 P19784 1/20 0.41
CSNK2A1 P68400 1/20 0.41
KDM5A P29375 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3333875 0.77 NR1H4 (0.46) RXRARXRBRXRGPSEN1PSEN2
SCHEMBL693269 0.77 SRD5A2 (0.90) SRD5A2CYP2C8RXRARXRBRXRG
SCHEMBL5023264 0.76 TNIK (0.46) MAPK1MAP2K4MAPK6MAPKAPK3KMT2A
SCHEMBL69008 0.74 MEN1 (0.50) MAPK1MAP2K4MAPK6MAPKAPK3MAPKAPK5
SCHEMBL28936490 0.74 SRD5A2 (0.57) SRD5A2CYP2C8MEN1LMNAKMT2A
SCHEMBL5022735 0.73 TNIK (0.43) KMT2A
SCHEMBL26477869 0.72 RAF1 (0.55) MAPK1MAP2K4MAPK6MAPKAPK3MAPKAPK5
SCHEMBL28775522 0.72 HTR2C (0.45)
SCHEMBL505133 0.72 SRD5A2 (0.77) SRD5A2MAPK1MAP2K4MAPK6MAPKAPK3
SCHEMBL30737531 0.71 HDAC1 (0.54) PPARAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150958-A1 SUBSTITUTED PYRAZOLE CARBOXYLIC ACIDS USED TO COMBAT ANAEMIAS Bayer Aktiengesellschaft (DE) 2001-11-07 EP disclosed
WO-2000046208-A1 SUBSTITUTED PYRAZOLE CARBOXYLIC ACIDS USED TO COMBAT ANAEMIAS BAYER AKTIENGESELLSCHAFT (DE) 2000-08-10 WO disclosed