SCHEMBL505133

SCHEMBL505133

O=C(O)c1ccc(-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.77
RXRA P19793 2/20 0.75
RXRB P28702 2/20 0.75
RXRG P48443 2/20 0.75
CYP2C8 P10632 1/20 0.67
CES2 O00748 1/20 0.61
CES1 P23141 1/20 0.61
MAP4K4 O95819 1/20 0.60
BCL2L1 Q07817 1/20 0.59
BAD Q92934 1/20 0.59
EPHX2 P34913 1/20 0.59
KIF11 P52732 2/20 0.58
P2RY14 Q15391 2/20 0.57
SLC6A2 P23975 1/20 0.57
DHODH Q02127 1/20 0.55
MAPK1 P28482 2/20 0.54
MAP2K4 P45985 2/20 0.54
MAPK6 Q16659 2/20 0.54
MAPKAPK3 Q16644 1/20 0.54
MAPKAPK5 Q8IW41 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5313295 0.98 SRD5A2 (0.74) SRD5A2RXRARXRBRXRGCYP2C8
SCHEMBL78879 0.93 SRD5A2 (0.87) SRD5A2RXRARXRBRXRGCYP2C8
SCHEMBL1330891 0.93 SRD5A2 (0.87) SRD5A2RXRARXRBRXRGCYP2C8
SCHEMBL6762584 0.91 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGCYP2C8
Hydrochloric Acid SCHEMBL8432890 0.91 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGCYP2C8
SCHEMBL23521062 0.91 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGCYP2C8
Water SCHEMBL28138640 0.91 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGCYP2C8
SCHEMBL29208531 0.91 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGCYP2C8
SCHEMBL1042428 0.91 SRD5A2 (0.83) SRD5A2RXRARXRBRXRGCYP2C8
Ethylene SCHEMBL715322 0.89 SRD5A2 (0.80) SRD5A2RXRARXRBRXRGCYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 168 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2167077-A2 ARYL/HETARYLAMIDES AS MODULATORS OF THE EP2 RECEPTOR Bayer Schering Pharma Aktiengesellschaft (DE) 2010-03-31 EP claimed
US-20090023741-A1 ARYL/HETARYLAMIDES AS MODULATORS OF THE EP2 RECEPTOR BAYER SCHERING PHARMA AG (DE) 2009-01-22 US claimed
WO-2008152099-A2 ARYL/HETARYLAMIDES AS MODULATORS OF THE EP2 RECEPTOR BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-12-18 WO claimed
US-7368462-B1 Melanin concentrating hormone antagonists THE PROCTER & GAMBLE COMPANY (US) 2008-05-06 US claimed
US-7304065-B2 Melanin concentrating hormone antagonists THE PROCTER & GAMBLE COMPANY (US) 2007-12-04 US claimed
WO-2007044574-A2 PHARMACEUTICAL COMPOSITIONS, METHODS OF PREPARATION THEREOF, AND METHODS OF TREATMENT TRANSTECH PHARMA, INC. (US) 2007-04-19 WO claimed
US-20070082952-A1 Pharmaceutical compositions, methods of preparation thereof, and methods of treatment TRANSTECH PHARMA, INC. 2007-04-12 US claimed
EP-1667958-A2 MELANIN CONCENTRATING HORMONE ANTAGONISTS THE PROCTER & GAMBLE COMPANY (US) 2006-06-14 EP claimed
WO-2005033063-A2 MELANIN CONCENTRATING HORMONE ANTAGONISTS THE PROCTER & GAMBLE COMPANY (US) 2005-04-14 WO claimed
US-20050075324-A1 Melanin concentrating hormone antagonists THE PROCTER & GAMBLE COMPANY (US) 2005-04-07 US claimed
US-20040147557-A1 Aryl piperidine derivatives as inducers of ldl-receptor expression BOUILLOT ANNE (FR) 2004-07-29 US claimed
US-20040077654-A1 Aryl piperidine and piperazine derivatives as inducers of ldl-receptor expression SMITHKLINE BEECHAM CORPORATION 2004-04-22 US claimed
EP-1351937-A1 ARYL PIPERIDINE DERIVATIVES AS INDUCERS OF LDL-RECEPTOR EXPRESSION GLAXO GROUP LIMITED (GB) 2003-10-15 EP claimed
EP-1351936-A1 ARYL PIPERIDINE AND PIPERAZINE DERIVATIVES AS INDUCERS OF LDL-RECEPTOR EXPRESSION GLAXO GROUP LIMITED (GB) 2003-10-15 EP claimed
WO-2002055496-A1 ARYL PIPERIDINE AND PIPERAZINE DERIVATIVES AS INDUCERS OF LDL-RECEPTOR EXPRESSION GLAXO GROUP LIMITED (GB) 2002-07-18 WO claimed
WO-2002055497-A1 ARYL PIPERIDINE DERIVATIVES AS INDUCERS OF LDL-RECEPTOR EXPRESSION GLAXO GROUP LIMITED (GB) 2002-07-18 WO claimed
US-20250346585-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS ALEXION PHARMACEUTICALS, INC. (US) 2025-11-13 US disclosed
US-20250179046-A1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS ZOETIS SERVICES LLC 2025-06-05 US disclosed
EP-1026149-A1 AMIDOCARBOXYLIC ACID DERIVATIVES Sankyo Company Limited (JP) 2000-08-09 EP disclosed
EP-0341514-A2 Process for the preparation of asymmetrical biaryle compounds BAYER AG (DE) 1989-11-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250179046-A1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS HTR2B, HTR1B, HTR5A SRD5A2 2082/4885RXRA 3714/4885RXRB 2415/4885
US-20050075324-A1 Melanin concentrating hormone antagonists MCHR1, MCHR2, MC1R SRD5A2 671/4885RXRA 1395/4885RXRB 1565/4885
US-20250346585-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS C5, C1S, C9 SRD5A2 2235/4885RXRA 4456/4885RXRB 4252/4885
US-20090023741-A1 ARYL/HETARYLAMIDES AS MODULATORS OF THE EP2 RECEPTOR PTGER2, PTGER1, PTGDR2 SRD5A2 447/4885RXRA 378/4885RXRB 394/4885
US-20040147557-A1 Aryl piperidine derivatives as inducers of ldl-receptor expression NR1H2, NR1H3, NR1H4 SRD5A2 303/4885RXRA 53/4885RXRB 66/4885
US-20040077654-A1 Aryl piperidine and piperazine derivatives as inducers of ldl-receptor expression LDLR, NR1H2, NCOR1 SRD5A2 3206/4885RXRA 139/4885RXRB 121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.