SCHEMBL7848426

SCHEMBL7848426

O=C(O)C(=O)Nc1ccc(O)cc1C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.69
PTPRC P08575 2/20 0.69
PTPN2 P17706 2/20 0.69
PTPRB P23467 2/20 0.69
PTPRE P23469 2/20 0.69
PTPN6 P29350 2/20 0.69
PTPRA P18433 1/20 0.69
KMT2A Q03164 5/20 0.57
ALDH1A1 P00352 5/20 0.57
MAPT P10636 4/20 0.57
MEN1 O00255 4/20 0.57
TDP1 Q9NUW8 3/20 0.57
HTT P42858 1/20 0.57
LMNA P02545 1/20 0.54
RAB9A P51151 1/20 0.54
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11494815 0.83 PTPN1 (0.67) PTPN1PTPRCPTPN2PTPRBPTPRE
SCHEMBL5409391 0.82 TDP1 (0.55) PTPN1PTPRCPTPN2PTPRBPTPRE
SCHEMBL7989039 0.81 PTPN1 (1.00) PTPN1PTPRCPTPN2PTPRBPTPRE
SCHEMBL7988908 0.81 KDM4E (0.70) PTPN1PTPRCPTPN2PTPRBPTPRE
SCHEMBL7850074 0.81 PTPN1 (0.65) PTPN1PTPRCPTPN2PTPRBPTPRE
SCHEMBL7836703 0.81 PTPN1 (0.65) PTPN1PTPRCPTPN2PTPRBPTPRE
SCHEMBL31451940 0.81 KDM4E (0.69) KMT2AALDH1A1MAPTMEN1TDP1
SCHEMBL28253565 0.81 KMT2A (0.57) PTPN1PTPRCPTPN2PTPRBPTPRE
SCHEMBL8533041 0.81 KDM4E (0.69) KMT2AALDH1A1MAPTMEN1TDP1
SCHEMBL20466337 0.80 CA12 (0.57) PTPN1PTPRCPTPN2PTPRBPTPRE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1062199-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPASES) NOVO NORDISK A/S (DK) 2000-12-27 EP claimed
WO-1999046236-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPASES) NOVO NORDISK A/S (DK) 1999-09-16 WO claimed
US-6225329-B1 USEFUL IN THE TREATMENT OF TYPE I DIABETES, TYPE II DIABETES, IMPAIRED GLUCOSE TOLERANCE, INSULIN AUTOIMMUNITY DISEASES WITH DYSFUNCTIONS OF THE COAGULATION SYSTEM, ALLERGIC DISEASES NOVO NORDISK A/S (DK) 2001-05-01 US disclosed
EP-1080068-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES Novo Nordisk A/S (DK) 2001-03-07 EP disclosed
EP-1062199-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPASES) NOVO NORDISK A/S (DK) 2000-12-27 EP disclosed
WO-1999046237-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES NOVO NORDISK A/S (DK) 1999-09-16 WO disclosed
WO-1999046236-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPASES) NOVO NORDISK A/S (DK) 1999-09-16 WO disclosed