SCHEMBL7849562

SCHEMBL7849562

O=C1CC2(CCN(CCc3cccc4ccccc34)CC2)Oc2ccc(NS(=O)(=O)c3ccccc3)cc21

nearest known ligand 0.80

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 9/20 0.80
ADRA1A P35348 8/20 0.80
ADRA1B P35368 8/20 0.80
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852948 0.86 ADRA1D (1.00) ADRA1DADRA1AADRA1BKCNH2
SCHEMBL7848678 0.83 ADRA1D (1.00) ADRA1DADRA1AADRA1BKCNH2
SCHEMBL7845026 0.82 ADRA1D (0.78) ADRA1DADRA1AADRA1B
SCHEMBL7851129 0.80 ADRA1D (0.75) ADRA1DADRA1AADRA1B
SCHEMBL7849708 0.77 ADRA1D (0.65) ADRA1DADRA1AADRA1BKCNH2
SCHEMBL8568967 0.73 KCNH2 (0.79) ADRA1DADRA1AADRA1BKCNH2
SCHEMBL9451723 0.72 ADRA1D (1.00) ADRA1DADRA1AADRA1BKCNH2
Hydrochloric Acid SCHEMBL8565725 0.72 ADRA1D (0.98) ADRA1DADRA1AADRA1BKCNH2
SCHEMBL7849561 0.71 ADRA1D (0.44) ADRA1DADRA1AADRA1B
SCHEMBL8569268 0.71 ADRA1D (0.70) ADRA1DADRA1AADRA1BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0831824-A4 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2001-05-02 EP disclosed
EP-0831824-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-04-01 EP disclosed
WO-1996039140-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-12-12 WO disclosed