SCHEMBL7853124

SCHEMBL7853124

N[C@@H]1C=CC[C@@H]2CN(c3ncc4c(=O)c(C(=O)O)cn(C5CC5F)c4c3Cl)C[C@@H]21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
POLB P06746 2/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
CYP3A4 P08684 3/20 0.36
DPP4 P27487 5/20 0.34
CYP2C9 P11712 2/20 0.33
EPHA2 P29317 1/20 0.33
FLT4 P35916 1/20 0.33
GSK3B P49841 1/20 0.33
RARB P10826 1/20 0.33
TBXAS1 P24557 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
HPGD P15428 1/20 0.30
XBP1 P17861 1/20 0.30
NFKB1 P19838 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852626 1.00 ALDH1A1 (0.38) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL8695749 1.00 ALDH1A1 (0.38) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7853126 0.90
SCHEMBL7852422 0.89 POLB (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL8697881 0.89 CYP3A4 (0.35) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7841699 0.89 CYP3A4 (0.35) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL8695363 0.88 ALDH1A1 (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1
Bromide SCHEMBL8693293 0.88 ALDH1A1 (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL8693387 0.86 ALDH1A1 (0.39) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL7851219 0.86 ALDH1A1 (0.39) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726270-B1 Derivatives of 1,6-naphthyridone carboxylic acids BAYER AG (DE) 2001-05-23 EP disclosed
EP-0726270-A1 Derivatives of 1,6-naphthyridine carboxylic acids BAYER AG (DE) 1996-08-14 EP disclosed