SCHEMBL7854584

SCHEMBL7854584

COc1cc2c(cc1Br)CCN(CCCC(CCCC(=O)CCc1ccc(F)cc1)(c1ccccc1)c1ccccc1)C2C1CCC1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.39
LMNA P02545 1/20 0.39
MTNR1B P49286 6/20 0.37
MTNR1A P48039 1/20 0.37
ALOX5 P09917 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
HCRTR1 O43613 2/20 0.35
HCRTR2 O43614 2/20 0.35
RXFP1 Q9HBX9 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TSHR P16473 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7855411 1.00 TP53 (0.39) TP53LMNAMTNR1BMTNR1AALOX5
SCHEMBL7854768 0.93 TP53 (0.38) TP53LMNAMTNR1BALOX5HDAC3
Hydrochloric Acid SCHEMBL7854514 0.93 TP53 (0.38) TP53LMNAMTNR1BALOX5HDAC3
Hydrochloric Acid SCHEMBL7854779 0.93 TP53 (0.42) TP53LMNAMTNR1BHCRTR1HCRTR2
Hydrochloric Acid SCHEMBL7847146 0.91 HCRTR1 (0.40) TP53LMNAMTNR1BMTNR1AHDAC3
Hydrochloric Acid SCHEMBL7845209 0.90 LMNA (0.40) TP53LMNAMTNR1BMTNR1AALOX5
SCHEMBL7838649 0.89 LMNA (0.41) TP53LMNAMTNR1BMTNR1AALOX5
Hydrochloric Acid SCHEMBL7855697 0.87 LMNA (0.40) TP53LMNAMTNR1BMTNR1AALOX5
Hydrochloric Acid SCHEMBL7847363 0.85 HCRTR1 (0.46) TP53LMNAMTNR1BHCRTR1HCRTR2
Hydrochloric Acid SCHEMBL7853340 0.84 HCRTR1 (0.41) TP53LMNAMTNR1BHDAC3HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129076-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AS LHRH ANTAGONISTS ABBOTT LABORATORIES (US) 2001-09-05 EP disclosed
WO-2000029380-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AS LHRH ANTAGONISTS ABBOTT LABORATORIES (US) 2000-05-25 WO disclosed
US-5981521-A USEFUL FOR TREATING VARIOUS HORMONE DEPENDENT DISEASES, INCLUDING PROSTATE CANCER, ENDOMETRIOSIS, UTERINE FIBROIDS, PRECOCIOUS PUBERTY, BENIGN PROSTATE HYPERTROPY AND IN VITRO FERTILIZATION ABBOTT LABORATORIES (US) 1999-11-09 US disclosed