SCHEMBL7855595

SCHEMBL7855595

Cc1c(C)c2c(c(C)c1O)CCC(C)(C(=O)NCCc1ccc(NC(=N)Cc3cccs3)cc1)O2

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 18/20 0.47
BCHE P06276 17/20 0.47
MAOB P27338 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856139 0.92 ACHE (0.47) ACHEBCHEMAOBPTGS1PTGS2
SCHEMBL4401509 0.88 ACHE (0.46) ACHEBCHEMAOBPTGS1PTGS2
Hydrochloric Acid SCHEMBL4411888 0.88 ACHE (0.45) ACHEBCHEMAOBPTGS1PTGS2
SCHEMBL9312837 0.81 PTGS1 (0.55) ACHEBCHEMAOBPTGS1PTGS2
SCHEMBL2058864 0.81 PTGS1 (0.60) ACHEBCHEMAOBPTGS1PTGS2
SCHEMBL4412022 0.81 ACHE (0.46) ACHEBCHEMAOBPTGS1PTGS2
Hydrochloric Acid SCHEMBL4396247 0.80 ACHE (0.45) ACHEBCHEMAOBPTGS1PTGS2
SCHEMBL2059364 0.80 PTGS1 (0.58) ACHEBCHEMAOBPTGS1PTGS2
Hydrochloric Acid SCHEMBL4491799 0.80 ACHE (0.44) ACHEBCHEMAOBPTGS1PTGS2
SCHEMBL4319066 0.78 PTGS1 (0.49) ACHEBCHEMAOBPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115719-A2 NOVEL AMIDINE DERIVATIVES, THEIR PREPARATION AND APPLICATION AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2001-07-18 EP disclosed
WO-2000017190-A2 AMIDINE DERIVATIVES, THEIR PREPARATION AND APPLICATION AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2000-03-30 WO disclosed