SCHEMBL7856003

SCHEMBL7856003

CCc1ccc(-c2nc(N)ncc2-c2ncc[nH]2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
ADORA1 P30542 10/20 0.41
ADORA2A P29274 6/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
RPS6KA3 P51812 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NISCH Q9Y2I1 1/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MEN1 O00255 1/20 0.37
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
P2RX3 P56373 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7023035 0.78 CYP1A2 (0.39) ADORA1ADORA2ASMN1; SMN2CYP1A2CYP3A4
SCHEMBL7855999 0.77 ASIC3 (0.44) KMT2AADORA1ADORA2ASMN1; SMN2RPS6KA3
SCHEMBL15587042 0.75 NISCH (0.63) ADORA1ADORA2ACYP1A2CYP3A4CYP2D6
SCHEMBL7856164 0.71 CSNK1A1 (0.43) KMT2AADORA1ADORA2ANISCH
SCHEMBL4971068 0.71 MAP3K14 (0.49) KMT2AADORA1ADORA2ALMNAMAPT
SCHEMBL7853495 0.71 GSK3B (0.46)
SCHEMBL7023251 0.71 GSK3B (0.46)
SCHEMBL5089143 0.71 GSK3B (0.52)
SCHEMBL4972846 0.70 GSK3B (0.52) KMT2AADORA1ADORA2ARPS6KA3LMNA
SCHEMBL27559815 0.68 GSK3B (0.42) KMT2AADORA1CYP1A2MEN1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1312807-A Inhibitors of glycogen synthase kinase 3 CHIRON CORP (US) 2001-09-12 CN disclosed
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed