SCHEMBL7856232

SCHEMBL7856232

NC(=O)Nc1cccc(C(=O)Nc2cccc(C(CC(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 5/20 0.50
KCNK9 Q9NPC2 4/20 0.50
ITGB3 P05106 2/20 0.50
ITGA2B P08514 2/20 0.50
KMT2A Q03164 5/20 0.47
POLB P06746 2/20 0.47
MEN1 O00255 4/20 0.47
PARP1 P09874 2/20 0.46
PARP10 Q53GL7 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.46
RAB9A P51151 2/20 0.46
NPC1 O15118 2/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SIRT1 Q96EB6 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856433 0.90 ITGB3 (0.54) KCNK3KCNK9ITGB3ITGA2BKMT2A
SCHEMBL7856436 0.85 ITGB3 (0.48) KCNK3KCNK9ITGB3ITGA2BKMT2A
SCHEMBL7856438 0.84 CASR (0.49) KCNK3KCNK9KMT2APOLBMEN1
SCHEMBL7455765 0.84 ITGB3 (0.58) KCNK3KCNK9ITGB3ITGA2BKMT2A
SCHEMBL2839379 0.82 MAPK1 (0.55) KCNK3KCNK9ITGB3ITGA2BKMT2A
SCHEMBL2837451 0.82 ITGB3 (0.62) KCNK3KCNK9ITGB3ITGA2B
SCHEMBL2838433 0.81 ITGB3 (0.60) ITGB3ITGA2BKMT2APOLBMEN1
SCHEMBL2836646 0.81 MEN1 (0.47) KCNK3KCNK9ITGB3ITGA2BKMT2A
SCHEMBL2833499 0.81 KMT2A (0.53) KCNK3KCNK9ITGB3ITGA2BKMT2A
SCHEMBL2837526 0.80 KMT2A (0.49) ITGB3ITGA2BKMT2APOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed