SCHEMBL7856993

SCHEMBL7856993

N#Cc1ccc(-c2ccc3c(c2)C[C@@]2(CCN4CCCC[C@H]4C2)O3)cc1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 15/20 0.40
KCNH2 Q12809 3/20 0.40
MCHR1 Q99705 2/20 0.38
OTUD7B Q6GQQ9 1/20 0.37
CYP2D6 P10635 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856996 1.00 HRH3 (0.40) HRH3KCNH2MCHR1OTUD7BCYP2D6
SCHEMBL7858469 1.00 HRH3 (0.40) HRH3KCNH2MCHR1OTUD7BCYP2D6
SCHEMBL7856633 1.00 HRH3 (0.40) HRH3KCNH2MCHR1OTUD7BCYP2D6
SCHEMBL863982 1.00 HRH3 (0.40) HRH3KCNH2MCHR1OTUD7BCYP2D6
SCHEMBL863601 0.97 HRH3 (0.40) HRH3KCNH2OTUD7BCYP2D6
SCHEMBL863414 0.96 HRH3 (0.38) HRH3KCNH2MCHR1OTUD7B
SCHEMBL863725 0.93 OTUD7B (0.37) HRH3KCNH2MCHR1OTUD7B
SCHEMBL863544 0.92 HRH3 (0.42) HRH3KCNH2CYP2D6
SCHEMBL863455 0.92 KCNH2 (0.45) HRH3KCNH2CYP2D6
SCHEMBL864143 0.92 HRH3 (0.44) HRH3KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010144571-A1 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2010-12-16 WO disclosed